PDB Information

PDB4ZYQ
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli
Gene SourcePlasmodium falciparum FcB1/Columbia
Primary Citation
Potent dual inhibitors of Plasmodium falciparum M1 and M17 aminopeptidases through optimization of S1 pocket interactions.
Drinkwater, N., Vinh, N.B., Mistry, S.N., Bamert, R.S., Ruggeri, C., Holleran, J.P., Loganathan, S., Paiardini, A., Charman, S.A., Powell, A.K., Avery, V.M., McGowan, S., Scammells, P.J.
Eur.J.Med.Chem.
HeaderHydrolase/Hydrolase Inhibitor
Released2015-05-22
Resolution2.600
CATH Insert Date10 Apr, 2016

PDB Images (37)

PDB Prints

PDB Chains (12)

Chain ID Date inserted into CATH CATH Status
A 11 Apr, 2016 Chopped
B 11 Apr, 2016 Chopped
C 11 Apr, 2016 Chopped
D 11 Apr, 2016 Chopped
E 11 Apr, 2016 Chopped
F 11 Apr, 2016 Chopped
G 11 Apr, 2016 Chopped
H 11 Apr, 2016 Chopped
I 11 Apr, 2016 Chopped
J 11 Apr, 2016 Chopped
K 11 Apr, 2016 Chopped
L 11 Apr, 2016 Chopped

CATH Domains (24)

Domain ID Date inserted into CATH Superfamily CATH Status
4zyqA01 03 May, 2016 3.40.220.10 Assigned
4zyqA02 03 May, 2016 3.40.630.10 Assigned
4zyqB01 03 May, 2016 3.40.220.10 Assigned
4zyqB02 03 May, 2016 3.40.630.10 Assigned
4zyqC01 03 May, 2016 3.40.220.10 Assigned
4zyqC02 03 May, 2016 3.40.630.10 Assigned
4zyqD01 03 May, 2016 3.40.220.10 Assigned
4zyqD02 03 May, 2016 3.40.630.10 Assigned
4zyqE01 03 May, 2016 3.40.220.10 Assigned
4zyqE02 03 May, 2016 3.40.630.10 Assigned
4zyqF01 03 May, 2016 3.40.220.10 Assigned
4zyqF02 03 May, 2016 3.40.630.10 Assigned
4zyqG01 03 May, 2016 3.40.220.10 Assigned
4zyqG02 03 May, 2016 3.40.630.10 Assigned
4zyqH01 03 May, 2016 3.40.220.10 Assigned
4zyqH02 03 May, 2016 3.40.630.10 Assigned
4zyqI01 03 May, 2016 3.40.220.10 Assigned
4zyqI02 03 May, 2016 3.40.630.10 Assigned
4zyqJ01 03 May, 2016 3.40.220.10 Assigned
4zyqJ02 03 May, 2016 3.40.630.10 Assigned
4zyqK01 03 May, 2016 3.40.220.10 Assigned
4zyqK02 03 May, 2016 3.40.630.10 Assigned
4zyqL01 03 May, 2016 3.40.220.10 Assigned
4zyqL02 03 May, 2016 3.40.630.10 Assigned

UniProtKB Entries (12)

Accession Gene ID Taxon Description
A0A024V0B1 A0A024V0B1_PLAFA Plasmodium falciparum Vietnam Oak-Knoll (FVO) Uncharacterized protein
A0A024V0B1 A0A024V0B1_PLAFA Plasmodium falciparum Vietnam Oak-Knoll (FVO) Uncharacterized protein
A0A024V0B1 A0A024V0B1_PLAFA Plasmodium falciparum Vietnam Oak-Knoll (FVO) Uncharacterized protein
A0A024V0B1 A0A024V0B1_PLAFA Plasmodium falciparum Vietnam Oak-Knoll (FVO) Uncharacterized protein
A0A024V0B1 A0A024V0B1_PLAFA Plasmodium falciparum Vietnam Oak-Knoll (FVO) Uncharacterized protein
A0A024V0B1 A0A024V0B1_PLAFA Plasmodium falciparum Vietnam Oak-Knoll (FVO) Uncharacterized protein
A0A024V0B1 A0A024V0B1_PLAFA Plasmodium falciparum Vietnam Oak-Knoll (FVO) Uncharacterized protein
A0A024V0B1 A0A024V0B1_PLAFA Plasmodium falciparum Vietnam Oak-Knoll (FVO) Uncharacterized protein
A0A024V0B1 A0A024V0B1_PLAFA Plasmodium falciparum Vietnam Oak-Knoll (FVO) Uncharacterized protein
A0A024V0B1 A0A024V0B1_PLAFA Plasmodium falciparum Vietnam Oak-Knoll (FVO) Uncharacterized protein
A0A024V0B1 A0A024V0B1_PLAFA Plasmodium falciparum Vietnam Oak-Knoll (FVO) Uncharacterized protein
A0A024V0B1 A0A024V0B1_PLAFA Plasmodium falciparum Vietnam Oak-Knoll (FVO) Uncharacterized protein