CATH Classification

Domain Context

CATH Clusters

Superfamily Retinoid X Receptor
Functional Family Peroxisome proliferator-activated receptor gamma

Enzyme Information

UniProtKB Entries (1)

P37231
PPARG_HUMAN
Homo sapiens
Peroxisome proliferator-activated receptor gamma

PDB Structure

PDB 5TTO
External Links
Method X-RAY DIFFRACTION
Organism
Primary Citation
Structure-Activity Relationship of 2,4-Dichloro-N-(3,5-dichloro-4-(quinolin-3-yloxy)phenyl)benzenesulfonamide (INT131) Analogs for PPAR gamma-Targeted Antidiabetics.
Frkic, R.L., He, Y., Rodriguez, B.B., Chang, M.R., Kuruvilla, D., Ciesla, A., Abell, A.D., Kamenecka, T.M., Griffin, P.R., Bruning, J.B.
J. Med. Chem.