CATH Classification

Domain Context

CATH Clusters

Superfamily Retinoid X Receptor
Functional Family Estrogen receptor

Enzyme Information

UniProtKB Entries (1)

P03372
ESR1_HUMAN
Homo sapiens
Estrogen receptor

PDB Structure

PDB 2IOK
External Links
Method X-RAY DIFFRACTION
Organism Escherichia
Primary Citation
Estrogen receptor ligands. Part 16: 2-Aryl indoles as highly subtype selective ligands for ERalpha
Dykstra, K.D., Guo, L., Birzin, E.T., Chan, W., Yang, Y.T., Hayes, E.C., DaSilva, C.A., Pai, L.-Y., Mosley, R.T., Kraker, B., Fitzgerald, P.M.D., DiNinno, F., Rohrer, S.P., Schaeffer, J.M., Hammond, M.L.
Bioorg.Med.Chem.Lett.