PDB Information

PDB6DQ9
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli
Gene SourceHomo sapiens
Primary Citation
Structure-Based Engineering of Irreversible Inhibitors against Histone Lysine Demethylase KDM5A.
Horton, J.R., Woodcock, C.B., Chen, Q., Liu, X., Zhang, X., Shanks, J., Rai, G., Mott, B.T., Jansen, D.J., Kales, S.C., Henderson, M.J., Cyr, M., Pohida, K., Hu, X., Shah, P., Xu, X., Jadhav, A., Maloney, D.J., Hall, M.D., Simeonov, A., Fu, H., Vertino, P.M., Cheng, X.
J. Med. Chem.
HeaderOxidoreductase/Inhibitor
Released2018-06-10
Resolution1.750
CATH Insert Date16 Dec, 2018

PDB Images (3)

PDB Prints

PDB Chains (1)

Chain ID Date inserted into CATH CATH Status
A 16 Dec, 2018 Chopped

CATH Domains (1)

Domain ID Date inserted into CATH Superfamily CATH Status
6dq9A00 28 Feb, 2019 2.60.120.650 Assigned

UniProtKB Entries (1)

Accession Gene ID Taxon Description
P29375 KDM5A_HUMAN Homo sapiens Lysine-specific demethylase 5A