PDB Information

PDB5VO4
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli-Pichia pastoris shuttle vector pPpARG4
Gene SourceHomo sapiens
Primary Citation
Structure-Based Approach To Identify 5-[4-Hydroxyphenyl]pyrrole-2-carbonitrile Derivatives as Potent and Tissue Selective Androgen Receptor Modulators.
Unwalla, R., Mousseau, J.J., Fadeyi, O.O., Choi, C., Parris, K., Hu, B., Kenney, T., Chippari, S., McNally, C., Vishwanathan, K., Kilbourne, E., Thompson, C., Nagpal, S., Wrobel, J., Yudt, M., Morris, C.A., Powell, D., Gilbert, A.M., Chekler, E.L.P.
J. Med. Chem.
HeaderHormone Receptor
Released2017-05-02
Resolution2.350
CATH Insert Date03 Jun, 2018

PDB Images (3)

PDB Prints

PDB Chains (1)

Chain ID Date inserted into CATH CATH Status
A 03 Jun, 2018 Chopped

CATH Domains (1)

Domain ID Date inserted into CATH Superfamily CATH Status
5vo4A00 28 Jun, 2018 1.10.565.10 Assigned

UniProtKB Entries (1)

Accession Gene ID Taxon Description
P10275 ANDR_HUMAN Homo sapiens Androgen receptor