CATH Classification

Domain Context

CATH Clusters

Superfamily Retinoid X Receptor
Functional Family Androgen receptor variant

Enzyme Information

UniProtKB Entries (1)

P10275
ANDR_HUMAN
Homo sapiens
Androgen receptor

PDB Structure

PDB 5VO4
External Links
Method X-RAY DIFFRACTION
Organism
Primary Citation
Structure-Based Approach To Identify 5-[4-Hydroxyphenyl]pyrrole-2-carbonitrile Derivatives as Potent and Tissue Selective Androgen Receptor Modulators.
Unwalla, R., Mousseau, J.J., Fadeyi, O.O., Choi, C., Parris, K., Hu, B., Kenney, T., Chippari, S., McNally, C., Vishwanathan, K., Kilbourne, E., Thompson, C., Nagpal, S., Wrobel, J., Yudt, M., Morris, C.A., Powell, D., Gilbert, A.M., Chekler, E.L.P.
J. Med. Chem.