PDB 5kby

PDB Information

PDB5KBY
MethodX-RAY DIFFRACTION
Host Organismunidentified baculovirus
Gene SourceHomo sapiens
Primary Citation
Trelagliptin (SYR-472, Zafatek), Novel Once-Weekly Treatment for Type 2 Diabetes, Inhibits Dipeptidyl Peptidase-4 (DPP-4) via a Non-Covalent Mechanism.
Grimshaw, C.E., Jennings, A., Kamran, R., Ueno, H., Nishigaki, N., Kosaka, T., Tani, A., Sano, H., Kinugawa, Y., Koumura, E., Shi, L., Takeuchi, K.
Plos One
HeaderHydrolase/Hydrolase Inhibitor
Released2016-06-03
Resolution2.240
CATH Insert Date24 Jul, 2016

PDB Images (13)

PDB Prints

PDB Chains (4)

Chain ID Date inserted into CATH CATH Status
A 25 Jul, 2016 Chopped
B 25 Jul, 2016 Chopped
C 25 Jul, 2016 Chopped
D 25 Jul, 2016 Chopped

CATH Domains (8)

Domain ID Date inserted into CATH Superfamily CATH Status
5kbyA01 01 Sep, 2016 2.140.10.30 Assigned
5kbyA02 01 Sep, 2016 3.40.50.1820 Assigned
5kbyB01 01 Sep, 2016 2.140.10.30 Assigned
5kbyB02 01 Sep, 2016 3.40.50.1820 Assigned
5kbyC01 01 Sep, 2016 2.140.10.30 Assigned
5kbyC02 01 Sep, 2016 3.40.50.1820 Assigned
5kbyD01 01 Sep, 2016 2.140.10.30 Assigned
5kbyD02 01 Sep, 2016 3.40.50.1820 Assigned

UniProtKB Entries (4)

Accession Gene ID Taxon Description
P27487 DPP4_HUMAN Homo sapiens Dipeptidyl peptidase 4
P27487 DPP4_HUMAN Homo sapiens Dipeptidyl peptidase 4
P27487 DPP4_HUMAN Homo sapiens Dipeptidyl peptidase 4
P27487 DPP4_HUMAN Homo sapiens Dipeptidyl peptidase 4