PDB Information

PDB5KBR
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli
Gene SourceHomo sapiens
Primary Citation
Optimization of Highly Kinase Selective Bis-anilino Pyrimidine PAK1 Inhibitors.
McCoull, W., Hennessy, E.J., Blades, K., Chuaqui, C., Dowling, J.E., Ferguson, A.D., Goldberg, F.W., Howe, N., Jones, C.R., Kemmitt, P.D., Lamont, G., Varnes, J.G., Ward, R.A., Yang, B.
ACS Med Chem Lett
HeaderTransferase
Released2016-06-03
Resolution2.360
CATH Insert Date09 Oct, 2016

PDB Images (7)

PDB Prints

PDB Chains (2)

Chain ID Date inserted into CATH CATH Status
A 10 Oct, 2016 Chopped
B 10 Oct, 2016 Chopped

CATH Domains (4)

Domain ID Date inserted into CATH Superfamily CATH Status
5kbrA01 15 Oct, 2016 3.30.200.20 Assigned
5kbrA02 15 Oct, 2016 1.10.510.10 Assigned
5kbrB01 15 Oct, 2016 3.30.200.20 Assigned
5kbrB02 15 Oct, 2016 1.10.510.10 Assigned

UniProtKB Entries (2)

Accession Gene ID Taxon Description
Q13153 PAK1_HUMAN Homo sapiens Serine/threonine-protein kinase PAK 1
Q13153 PAK1_HUMAN Homo sapiens Serine/threonine-protein kinase PAK 1