PDB Information

PDB5FH8
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli
Gene SourceHomo sapiens
Primary Citation
Identification and Development of 2,3-Dihydropyrrolo[1,2-a]quinazolin-5(1H)-one Inhibitors Targeting Bromodomains within the Switch/Sucrose Nonfermenting Complex.
Sutherell, C.L., Tallant, C., Monteiro, O.P., Yapp, C., Fuchs, J.E., Fedorov, O., Siejka, P., Muller, S., Knapp, S., Brenton, J.D., Brennan, P.E., Ley, S.V.
J.Med.Chem.
HeaderTranscription
Released2015-12-21
Resolution1.550
CATH Insert Date10 Jul, 2016

PDB Images (9)

PDB Prints

PDB Chains (4)

Chain ID Date inserted into CATH CATH Status
A 11 Jul, 2016 Chopped
B 11 Jul, 2016 Chopped
C 11 Jul, 2016 Chopped
D 11 Jul, 2016 Chopped

CATH Domains (4)

Domain ID Date inserted into CATH Superfamily CATH Status
5fh8A00 16 Jul, 2016 1.20.920.10 Assigned
5fh8B00 15 Jul, 2016 1.20.920.10 Assigned
5fh8C00 16 Jul, 2016 1.20.920.10 Assigned
5fh8D00 16 Jul, 2016 1.20.920.10 Assigned

UniProtKB Entries (4)

Accession Gene ID Taxon Description
Q86U86 PB1_HUMAN Homo sapiens Protein polybromo-1
Q86U86 PB1_HUMAN Homo sapiens Protein polybromo-1
Q86U86 PB1_HUMAN Homo sapiens Protein polybromo-1
Q86U86 PB1_HUMAN Homo sapiens Protein polybromo-1