PDB Information

PDB5ENQ
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli
Gene SourceEscherichia coli K-12
Primary Citation
Molecular basis for inhibition of AcrB multidrug efflux pump by novel and powerful pyranopyridine derivatives.
Sjuts, H., Vargiu, A.V., Kwasny, S.M., Nguyen, S.T., Kim, H.S., Ding, X., Ornik, A.R., Ruggerone, P., Bowlin, T.L., Nikaido, H., Pos, K.M., Opperman, T.J.
Proc.Natl.Acad.Sci.USA
HeaderTransport Protein
Released2015-11-09
Resolution1.800
CATH Insert Date17 Apr, 2016

PDB Images (25)

PDB Prints

PDB Chains (6)

Chain ID Date inserted into CATH CATH Status
A 18 Apr, 2016 Chopped
B 18 Apr, 2016 Chopped
C 18 Apr, 2016 Chopped
D 18 Apr, 2016 Chopped
E 18 Apr, 2016 Chopped
F 18 Apr, 2016 Chopped

CATH Domains (18)

Domain ID Date inserted into CATH Superfamily CATH Status
5enqA01 09 Jan, 2018 3.30.70.1430 Assigned
5enqA02 09 Jan, 2018 3.30.70.1320 Assigned
5enqA03 09 Jan, 2018 Holding pen
5enqA04 09 Jan, 2018 3.30.70.1430 Assigned
5enqA05 09 Jan, 2018 3.30.70.1440 Assigned
5enqB01 09 Jan, 2018 3.30.70.1430 Assigned
5enqB02 09 Jan, 2018 3.30.70.1320 Assigned
5enqB03 09 Jan, 2018 Holding pen
5enqB04 09 Jan, 2018 3.30.70.1430 Assigned
5enqB05 09 Jan, 2018 3.30.70.1440 Assigned
5enqC01 09 Jan, 2018 3.30.70.1430 Assigned
5enqC02 09 Jan, 2018 3.30.70.1320 Assigned
5enqC03 09 Jan, 2018 Holding pen
5enqC04 09 Jan, 2018 3.30.70.1430 Assigned
5enqC05 09 Jan, 2018 3.30.70.1440 Assigned
5enqD00 30 Nov, 2016 1.25.40.20 Assigned
5enqE00 30 Nov, 2016 1.25.40.20 Assigned
5enqF00 30 Nov, 2016 1.25.40.20 Assigned

UniProtKB Entries (3)

Accession Gene ID Taxon Description
P31224 ACRB_ECOLI Escherichia coli K-12 Multidrug efflux pump subunit AcrB
P31224 ACRB_ECOLI Escherichia coli K-12 Multidrug efflux pump subunit AcrB
P31224 ACRB_ECOLI Escherichia coli K-12 Multidrug efflux pump subunit AcrB