PDB Information

PDB5EJV
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli
Gene SourceHomo sapiens
Primary Citation
Discovery of biaryls as ROR gamma inverse agonists by using structure-based design.
Enyedy, I.J., Powell, N.A., Caravella, J., van Vloten, K., Chao, J., Banerjee, D., Marcotte, D., Silvian, L., McKenzie, A., Hong, V.S., Fontenot, J.D.
Bioorg.Med.Chem.Lett.
HeaderTranscription
Released2015-11-02
Resolution2.580
CATH Insert Date08 May, 2016

PDB Images (7)

PDB Prints

PDB Chains (4)

Chain ID Date inserted into CATH CATH Status
A 09 May, 2016 Chopped
B 09 May, 2016 Chopped
C 09 May, 2016 Rejected
D 09 May, 2016 Rejected

CATH Domains (2)

Domain ID Date inserted into CATH Superfamily CATH Status
5ejvA00 15 Jul, 2016 1.10.565.10 Assigned
5ejvB00 15 Jul, 2016 1.10.565.10 Assigned

UniProtKB Entries (2)

Accession Gene ID Taxon Description
P51449 RORG_HUMAN Homo sapiens Nuclear receptor ROR-gamma
P51449 RORG_HUMAN Homo sapiens Nuclear receptor ROR-gamma