CATH Classification

Domain Context

CATH Clusters

Superfamily Retinoid X Receptor
Functional Family Nuclear orphan receptor ROR-beta

Enzyme Information

UniProtKB Entries (1)

P51449
RORG_HUMAN
Homo sapiens
Nuclear receptor ROR-gamma

PDB Structure

PDB 5EJV
External Links
Method X-RAY DIFFRACTION
Organism
Primary Citation
Discovery of biaryls as ROR gamma inverse agonists by using structure-based design.
Enyedy, I.J., Powell, N.A., Caravella, J., van Vloten, K., Chao, J., Banerjee, D., Marcotte, D., Silvian, L., McKenzie, A., Hong, V.S., Fontenot, J.D.
Bioorg.Med.Chem.Lett.