PDB Information

PDB5DRB
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli
Gene SourceRattus norvegicus
Primary Citation
Small-molecule WNK inhibition regulates cardiovascular and renal function.
Yamada, K., Park, H.M., Rigel, D.F., DiPetrillo, K., Whalen, E.J., Anisowicz, A., Beil, M., Berstler, J., Brocklehurst, C.E., Burdick, D.A., Caplan, S.L., Capparelli, M.P., Chen, G., Chen, W., Dale, B., Deng, L., Fu, F., Hamamatsu, N., Harasaki, K., Herr, T., Hoffmann, P., Hu, Q.Y., Huang, W.J., Idamakanti, N., Imase, H., Iwaki, Y., Jain, M., Jeyaseelan, J., Kato, M., Kaushik, V.K., Kohls, D., Kunjathoor, V., LaSala, D., Lee, J., Liu, J., Luo, Y., Ma, F., Mo, R., Mowbray, S., Mogi, M., Ossola, F., Pandey, P., Patel, S.J., Raghavan, S., Salem, B., Shanado, Y.H., Trakshel, G.M., Turner, G., Wakai, H., Wang, C., Weldon, S., Wielicki, J.B., Xie, X., Xu, L., Yagi, Y.I., Yasoshima, K., Yin, J., Yowe, D., Zhang, J.H., Zheng, G., Monovich, L.
Nat.Chem.Biol.
HeaderTransferase/Transferase Inhibitor
Released2015-09-15
Resolution1.650
CATH Insert Date09 Oct, 2016

PDB Images (4)

PDB Prints

PDB Chains (1)

Chain ID Date inserted into CATH CATH Status
A 10 Oct, 2016 Chopped

CATH Domains (2)

Domain ID Date inserted into CATH Superfamily CATH Status
5drbA01 13 Oct, 2016 3.30.200.20 Assigned
5drbA02 13 Oct, 2016 1.10.510.10 Assigned

UniProtKB Entries (1)

Accession Gene ID Taxon Description
Q9JIH7 WNK1_RAT Rattus norvegicus Serine/threonine-protein kinase WNK1