PDB 5dey
PDB Information
PDB | 5DEY |
Method | X-RAY DIFFRACTION |
Host Organism | Escherichia coli |
Gene Source | Homo sapiens |
Primary Citation | Design of Selective PAK1 Inhibitor G-5555: Improving Properties by Employing an Unorthodox Low-pK a Polar Moiety.
Acs Med.Chem.Lett.
|
Header | Transferase/Transferase Inhibitor |
Released | 2015-08-26 |
Resolution | 2.100 |
CATH Insert Date | 10 Apr, 2016 |
PDB Images (7)
PDB Prints
PDB Chains (2)
Chain ID | Date inserted into CATH | CATH Status |
---|---|---|
A | 11 Apr, 2016 | Chopped |
B | 11 Apr, 2016 | Chopped |
CATH Domains (4)
Domain ID | Date inserted into CATH | Superfamily | CATH Status |
---|---|---|---|
5deyA01 | 07 May, 2016 | 3.30.200.20 | Assigned |
5deyA02 | 07 May, 2016 | 1.10.510.10 | Assigned |
5deyB01 | 07 May, 2016 | 3.30.200.20 | Assigned |
5deyB02 | 07 May, 2016 | 1.10.510.10 | Assigned |
UniProtKB Entries (2)
Accession | Gene ID | Taxon | Description |
---|---|---|---|
Q13153 | PAK1_HUMAN | Homo sapiens | Serine/threonine-protein kinase PAK 1 |
Q13153 | PAK1_HUMAN | Homo sapiens | Serine/threonine-protein kinase PAK 1 |