PDB Information

PDB4K3N
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli
Gene SourcePlasmodium falciparum 3D7
Primary Citation
Synthesis and Structure-Activity Relationships of Phosphonic Arginine Mimetics as Inhibitors of the M1 and M17 Aminopeptidases from Plasmodium falciparum.
Kannan Sivaraman, K., Paiardini, A., Sienczyk, M., Ruggeri, C., Oellig, C.A., Dalton, J.P., Scammells, P.J., Drag, M., McGowan, S.
J.Med.Chem.
HeaderHydrolase/Hydrolase Inhibitor
Released2013-04-11
Resolution2.000
CATH Insert Date07 Jul, 2013

PDB Images (37)

PDB Prints

PDB Chains (12)

Chain ID Date inserted into CATH CATH Status
A 08 Jul, 2013 Chopped
B 08 Jul, 2013 Chopped
C 08 Jul, 2013 Chopped
D 08 Jul, 2013 Chopped
E 08 Jul, 2013 Chopped
F 08 Jul, 2013 Chopped
G 08 Jul, 2013 Chopped
H 08 Jul, 2013 Chopped
I 08 Jul, 2013 Chopped
J 08 Jul, 2013 Chopped
K 08 Jul, 2013 Chopped
L 08 Jul, 2013 Chopped

CATH Domains (24)

Domain ID Date inserted into CATH Superfamily CATH Status
4k3nA01 09 Aug, 2013 3.40.220.10 Assigned
4k3nA02 09 Aug, 2013 3.40.630.10 Assigned
4k3nB01 09 Aug, 2013 3.40.220.10 Assigned
4k3nB02 09 Aug, 2013 3.40.630.10 Assigned
4k3nC01 09 Aug, 2013 3.40.220.10 Assigned
4k3nC02 09 Aug, 2013 3.40.630.10 Assigned
4k3nD01 09 Aug, 2013 3.40.220.10 Assigned
4k3nD02 09 Aug, 2013 3.40.630.10 Assigned
4k3nE01 09 Aug, 2013 3.40.220.10 Assigned
4k3nE02 09 Aug, 2013 3.40.630.10 Assigned
4k3nF01 09 Aug, 2013 3.40.220.10 Assigned
4k3nF02 09 Aug, 2013 3.40.630.10 Assigned
4k3nG01 09 Aug, 2013 3.40.220.10 Assigned
4k3nG02 09 Aug, 2013 3.40.630.10 Assigned
4k3nH01 09 Aug, 2013 3.40.220.10 Assigned
4k3nH02 09 Aug, 2013 3.40.630.10 Assigned
4k3nI01 09 Aug, 2013 3.40.220.10 Assigned
4k3nI02 09 Aug, 2013 3.40.630.10 Assigned
4k3nJ01 09 Aug, 2013 3.40.220.10 Assigned
4k3nJ02 09 Aug, 2013 3.40.630.10 Assigned
4k3nK01 09 Aug, 2013 3.40.220.10 Assigned
4k3nK02 09 Aug, 2013 3.40.630.10 Assigned
4k3nL01 09 Aug, 2013 3.40.220.10 Assigned
4k3nL02 09 Aug, 2013 3.40.630.10 Assigned

UniProtKB Entries (12)

Accession Gene ID Taxon Description
Q8IL11 Q8IL11_PLAF7 Plasmodium falciparum 3D7 M17 leucyl aminopeptidase
Q8IL11 Q8IL11_PLAF7 Plasmodium falciparum 3D7 M17 leucyl aminopeptidase
Q8IL11 Q8IL11_PLAF7 Plasmodium falciparum 3D7 M17 leucyl aminopeptidase
Q8IL11 Q8IL11_PLAF7 Plasmodium falciparum 3D7 M17 leucyl aminopeptidase
Q8IL11 Q8IL11_PLAF7 Plasmodium falciparum 3D7 M17 leucyl aminopeptidase
Q8IL11 Q8IL11_PLAF7 Plasmodium falciparum 3D7 M17 leucyl aminopeptidase
Q8IL11 Q8IL11_PLAF7 Plasmodium falciparum 3D7 M17 leucyl aminopeptidase
Q8IL11 Q8IL11_PLAF7 Plasmodium falciparum 3D7 M17 leucyl aminopeptidase
Q8IL11 Q8IL11_PLAF7 Plasmodium falciparum 3D7 M17 leucyl aminopeptidase
Q8IL11 Q8IL11_PLAF7 Plasmodium falciparum 3D7 M17 leucyl aminopeptidase
Q8IL11 Q8IL11_PLAF7 Plasmodium falciparum 3D7 M17 leucyl aminopeptidase
Q8IL11 Q8IL11_PLAF7 Plasmodium falciparum 3D7 M17 leucyl aminopeptidase