PDB Information

PDB4GV7
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli
Gene SourceHomo sapiens
Primary Citation
PARP Inhibitor with Selectivity Toward ADP-Ribosyltransferase ARTD3/PARP3
Lindgren, A.E.G., Karlberg, T., Thorsell, A.G., Hesse, M., Spjut, S., Ekblad, T., Andersson, C.D., Pinto, A.F., Weigelt, J., Hottiger, M.O., Linusson, A., Elofsson, M., Schuler, H.
Acs Chem.Biol.
HeaderTransferase/Transferase Inhibitor
Released2012-08-30
Resolution2.890
CATH Insert Date07 Jul, 2013

PDB Images (13)

PDB Prints

PDB Chains (4)

Chain ID Date inserted into CATH CATH Status
A 08 Jul, 2013 Chopped
B 08 Jul, 2013 Chopped
C 08 Jul, 2013 Chopped
D 08 Jul, 2013 Chopped

CATH Domains (8)

Domain ID Date inserted into CATH Superfamily CATH Status
4gv7A01 13 Sep, 2013 1.20.142.10 Assigned
4gv7A02 13 Sep, 2013 3.90.228.10 Assigned
4gv7B01 13 Sep, 2013 1.20.142.10 Assigned
4gv7B02 13 Sep, 2013 3.90.228.10 Assigned
4gv7C01 13 Sep, 2013 1.20.142.10 Assigned
4gv7C02 13 Sep, 2013 3.90.228.10 Assigned
4gv7D01 13 Sep, 2013 1.20.142.10 Assigned
4gv7D02 13 Sep, 2013 3.90.228.10 Assigned

UniProtKB Entries (4)

Accession Gene ID Taxon Description
P09874 PARP1_HUMAN Homo sapiens Poly [ADP-ribose] polymerase 1
P09874 PARP1_HUMAN Homo sapiens Poly [ADP-ribose] polymerase 1
P09874 PARP1_HUMAN Homo sapiens Poly [ADP-ribose] polymerase 1
P09874 PARP1_HUMAN Homo sapiens Poly [ADP-ribose] polymerase 1