PDB Information

PDB4FF8
MethodX-RAY DIFFRACTION
Host OrganismSpodoptera frugiperda
Gene SourceMus musculus
Primary Citation
Highly selective 2,4-diaminopyrimidine-5-carboxamide inhibitors of Sky kinase.
Powell, N.A., Hoffman, J.K., Ciske, F.L., Kaufman, M.D., Kohrt, J.T., Quin, J., Sheehan, D.J., Delaney, A., Baxi, S.M., Catana, C., McConnell, P., Ohren, J., Perrin, L.A., Edmunds, J.J.
Bioorg.Med.Chem.Lett.
HeaderTransferase/Transferase Inhibitor
Released2012-05-31
Resolution2.400
CATH Insert Date28 Mar, 2013

PDB Images (3)

PDB Prints

PDB Chains (1)

Chain ID Date inserted into CATH CATH Status
A 28 Mar, 2013 Chopped

CATH Domains (1)

Domain ID Date inserted into CATH Superfamily CATH Status
4ff8A00 14 Aug, 2013 1.10.510.10 Assigned

UniProtKB Entries (1)

Accession Gene ID Taxon Description
P55144 TYRO3_MOUSE Mus musculus Tyrosine-protein kinase receptor TYRO3