PDB Information

PDB3OCB
MethodX-RAY DIFFRACTION
Host OrganismSpodoptera frugiperda
Gene SourceHomo sapiens
Primary Citation
Discovery of pyrrolopyrimidine inhibitors of Akt.
Blake, J.F., Kallan, N.C., Xiao, D., Xu, R., Bencsik, J.R., Skelton, N.J., Spencer, K.L., Mitchell, I.S., Woessner, R.D., Gloor, S.L., Risom, T., Gross, S.D., Martinson, M., Morales, T.H., Vigers, G.P., Brandhuber, B.J.
Bioorg.Med.Chem.Lett.
HeaderTransferase
Released2010-08-09
Resolution2.700
CATH Insert Date19 Sep, 2010

PDB Images (9)

PDB Prints

PDB Chains (4)

Chain ID Date inserted into CATH CATH Status
A 20 Sep, 2010 Chopped
B 20 Sep, 2010 Chopped
C 20 Sep, 2010 Rejected
D 20 Sep, 2010 Rejected

CATH Domains (4)

Domain ID Date inserted into CATH Superfamily CATH Status
3ocbA01 30 Aug, 2013 3.30.200.20 Assigned
3ocbA02 30 Aug, 2013 1.10.510.10 Assigned
3ocbB01 29 Aug, 2013 3.30.200.20 Assigned
3ocbB02 29 Aug, 2013 1.10.510.10 Assigned

UniProtKB Entries (2)

Accession Gene ID Taxon Description
P31749 AKT1_HUMAN Homo sapiens RAC-alpha serine/threonine-protein kinase
P31749 AKT1_HUMAN Homo sapiens RAC-alpha serine/threonine-protein kinase