PDB 3o9v

PDB Information

PDB3O9V
MethodX-RAY DIFFRACTION
Host OrganismSpodoptera frugiperda
Gene SourceHomo sapiens
Primary Citation
Discovery of a 3-Pyridylacetic Acid Derivative (TAK-100) as a Potent, Selective and Orally Active Dipeptidyl Peptidase IV (DPP-4) Inhibitor.
Miyamoto, Y., Banno, Y., Yamashita, T., Fujimoto, T., Oi, S., Moritoh, Y., Asakawa, T., Kataoka, O., Yashiro, H., Takeuchi, K., Suzuki, N., Ikedo, K., Kosaka, T., Tsubotani, S., Tani, A., Sasaki, M., Funami, M., Amano, M., Yamamoto, Y., Aertgeerts, K., Yano, J., Maezaki, H.
J.Med.Chem.
HeaderHydrolase,Signaling Protein/Inhibitor
Released2010-08-04
Resolution2.750
CATH Insert Date13 Feb, 2011

PDB Images (13)

PDB Prints

PDB Chains (4)

Chain ID Date inserted into CATH CATH Status
A 14 Feb, 2011 Chopped
B 14 Feb, 2011 Chopped
C 14 Feb, 2011 Chopped
D 14 Feb, 2011 Chopped

CATH Domains (8)

Domain ID Date inserted into CATH Superfamily CATH Status
3o9vA01 18 Feb, 2011 2.140.10.30 Assigned
3o9vA02 18 Feb, 2011 3.40.50.1820 Assigned
3o9vB01 18 Feb, 2011 2.140.10.30 Assigned
3o9vB02 18 Feb, 2011 3.40.50.1820 Assigned
3o9vC01 18 Feb, 2011 2.140.10.30 Assigned
3o9vC02 18 Feb, 2011 3.40.50.1820 Assigned
3o9vD01 18 Feb, 2011 2.140.10.30 Assigned
3o9vD02 18 Feb, 2011 3.40.50.1820 Assigned

UniProtKB Entries (4)

Accession Gene ID Taxon Description
P27487 DPP4_HUMAN Homo sapiens Dipeptidyl peptidase 4
P27487 DPP4_HUMAN Homo sapiens Dipeptidyl peptidase 4
P27487 DPP4_HUMAN Homo sapiens Dipeptidyl peptidase 4
P27487 DPP4_HUMAN Homo sapiens Dipeptidyl peptidase 4