PDB Information

PDB3KF2
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli
Gene SourceHepatitis C virus
Primary Citation
Induced-Fit Binding of the Macrocyclic Noncovalent Inhibitor TMC435 to its HCV NS3/NS4A Protease Target
Cummings, M.D., Lindberg, J.D., Lin, T.-I., de Kock, H., Lenz, O., Lilja, E., Fellander, S., Baraznenok, V., Nystrom, S., Nilsson, M., Vrang, L., Edlund, M., Rosenquist, A., Samuelsson, B., Raboisson, P., Simmen, K.
Angew.Chem.Int.Ed.Engl.
HeaderHydrolase
Released2009-10-27
Resolution2.500
CATH Insert Date11 Mar, 2010

PDB Images (9)

PDB Prints

PDB Chains (4)

Chain ID Date inserted into CATH CATH Status
A 11 Mar, 2010 Chopped
B 11 Mar, 2010 Chopped
C 11 Mar, 2010 Rejected
D 11 Mar, 2010 Rejected

CATH Domains (4)

Domain ID Date inserted into CATH Superfamily CATH Status
3kf2A01 16 Apr, 2010 2.40.10.120 Assigned
3kf2A02 16 Apr, 2010 2.40.10.10 Assigned
3kf2B01 16 Apr, 2010 2.40.10.120 Assigned
3kf2B02 16 Apr, 2010 2.40.10.10 Assigned

UniProtKB Entries (4)

Accession Gene ID Taxon Description
B2Y2M9 B2Y2M9_9HEPC Hepacivirus C Genome polyprotein
Q6GYR8 Q6GYR8_9HEPC Hepacivirus C Genome polyprotein
B2Y2M9 B2Y2M9_9HEPC Hepacivirus C Genome polyprotein
Q6GYR8 Q6GYR8_9HEPC Hepacivirus C Genome polyprotein