PDB Information

PDB2RF2
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli
Gene SourceHIV-1 M:B_HXB2R
Primary Citation
Novel indole-3-sulfonamides as potent HIV non-nucleoside reverse transcriptase inhibitors (NNRTIs).
Zhao, Z., Wolkenberg, S.E., Lu, M., Munshi, V., Moyer, G., Feng, M., Carella, A.V., Ecto, L.T., Gabryelski, L.J., Lai, M.T., Prasad, S.G., Yan, Y., McGaughey, G.B., Miller, M.D., Lindsley, C.W., Hartman, G.D., Vacca, J.P., Williams, T.M.
Bioorg.Med.Chem.Lett.
HeaderTransferase
Released2007-09-27
Resolution2.400
CATH Insert Date03 Jan, 2008

PDB Images (12)

PDB Prints

PDB Chains (2)

Chain ID Date inserted into CATH CATH Status
A 03 Jan, 2008 Chopped
B 03 Jan, 2008 Chopped

CATH Domains (9)

Domain ID Date inserted into CATH Superfamily CATH Status
2rf2A01 04 Jan, 2008 3.10.10.10 Assigned
2rf2A02 04 Jan, 2008 3.30.70.270 Assigned
2rf2A03 04 Jan, 2008 3.30.70.270 Assigned
2rf2A04 04 Jan, 2008 3.30.70.270 Assigned
2rf2A05 04 Jan, 2008 3.30.420.10 Assigned
2rf2B01 04 Jan, 2008 3.10.10.10 Assigned
2rf2B02 04 Jan, 2008 3.30.70.270 Assigned
2rf2B03 04 Jan, 2008 3.30.70.270 Assigned
2rf2B04 04 Jan, 2008 3.30.70.270 Assigned

UniProtKB Entries (2)

Accession Gene ID Taxon Description
P04585 POL_HV1H2 HIV-1 M:B_HXB2R Gag-Pol polyprotein
P04585 POL_HV1H2 HIV-1 M:B_HXB2R Gag-Pol polyprotein