PDB Information

PDB2GTN
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli BL21(DE3)
Gene SourceMus musculus
Primary Citation
The development of novel C-2, C-8, and N-9 trisubstituted purines as inhibitors of TNF-alpha production.
Sabat, M., Vanrens, J.C., Clark, M.P., Brugel, T.A., Maier, J., Bookland, R.G., Laufersweiler, M.J., Laughlin, S.K., Golebiowski, A., De, B., Hsieh, L.C., Walter, R.L., Mekel, M.J., Janusz, M.J.
Bioorg.Med.Chem.Lett.
HeaderTransferase
Released2006-04-28
Resolution1.800
CATH Insert Date18 Jul, 2006

PDB Images (4)

PDB Prints

PDB Chains (1)

Chain ID Date inserted into CATH CATH Status
A 18 Jul, 2006 Chopped

CATH Domains (2)

Domain ID Date inserted into CATH Superfamily CATH Status
2gtnA01 17 Jul, 2007 3.30.200.20 Assigned
2gtnA02 17 Jul, 2007 1.10.510.10 Assigned

UniProtKB Entries (1)

Accession Gene ID Taxon Description
P47811 MK14_MOUSE Mus musculus Mitogen-activated protein kinase 14