PDB 6c2y
PDB Information
| PDB | 6C2Y |
| Method | X-RAY DIFFRACTION |
| Host Organism | Spodoptera aff. frugiperda 2 RZ-2014 |
| Gene Source | Homo sapiens |
| Primary Citation | Utilizing a structure-based docking approach to develop potent G protein-coupled receptor kinase (GRK) 2 and 5 inhibitors.
Bioorg. Med. Chem. Lett.
|
| Header | Transferase/Signaling Protein |
| Released | 2018-01-09 |
| Resolution | 2.740 |
| CATH Insert Date | 03 Jun, 2018 |
PDB Prints
PDB Chains (3)
| Chain ID | Date inserted into CATH | CATH Status |
|---|---|---|
| A | 03 Jun, 2018 | Chopped |
| B | 03 Jun, 2018 | Chopped |
| G | 03 Jun, 2018 | Chopped |
CATH Domains (7)
| Domain ID | Date inserted into CATH | Superfamily | CATH Status |
|---|---|---|---|
| 6c2yA01 | 28 Jun, 2018 | 1.10.287.1270 | Assigned |
| 6c2yA02 | 28 Jun, 2018 | 1.10.167.10 | Assigned |
| 6c2yA03 | 28 Jun, 2018 | 3.30.200.20 | Assigned |
| 6c2yA04 | 28 Jun, 2018 | 1.10.510.10 | Assigned |
| 6c2yA05 | 28 Jun, 2018 | 2.30.29.30 | Assigned |
| 6c2yB00 | 28 Jun, 2018 | 2.130.10.10 | Assigned |
| 6c2yG00 | 28 Jun, 2018 | 4.10.260.10 | Assigned |
UniProtKB Entries (3)
| Accession | Gene ID | Taxon | Description |
|---|---|---|---|
| P63212 | GBG2_BOVIN | Bos taurus | Guanine nucleotide-binding protein G(I)/G(S)/G(O) subunit gamma-2 |
| P62871 | GBB1_BOVIN | Bos taurus | Guanine nucleotide-binding protein G(I)/G(S)/G(T) subunit beta-1 |
| P25098 | ARBK1_HUMAN | Homo sapiens | Beta-adrenergic receptor kinase 1 |
