CATH Classification

Domain Context

CATH Clusters

Superfamily Retinoid X Receptor
Functional Family Nuclear orphan receptor ROR-beta

Enzyme Information

UniProtKB Entries (1)

P51449
RORG_HUMAN
Homo sapiens
Nuclear receptor ROR-gamma

PDB Structure

PDB 5LWP
External Links
Method X-RAY DIFFRACTION
Organism
Primary Citation
Discovery of phenoxyindazoles and phenylthioindazoles as ROR gamma inverse agonists.
Ouvry, G., Bouix-Peter, C., Ciesielski, F., Chantalat, L., Christin, O., Comino, C., Duvert, D., Feret, C., Harris, C.S., Lamy, L., Luzy, A.P., Musicki, B., Orfila, D., Pascau, J., Parnet, V., Perrin, A., Pierre, R., Polge, G., Raffin, C., Rival, Y., Taquet, N., Thoreau, E., Hennequin, L.F.
Bioorg.Med.Chem.Lett.