PDB Information

PDB6MAU
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli BL21(DE3)
Gene SourceHomo sapiens
Primary Citation
Lead optimization and efficacy evaluation of quinazoline-based BET family inhibitors for potential treatment of cancer and inflammatory diseases.
Yang, S.M., Yoshioka, M., Strovel, J.W., Urban, D.J., Hu, X., Hall, M.D., Jadhav, A., Maloney, D.J.
Bioorg. Med. Chem. Lett.
HeaderProtein Binding
Released2018-08-28
Resolution2.110
CATH Insert Date07 Apr, 2019

PDB Images (3)

PDB Prints

PDB Chains (1)

Chain ID Date inserted into CATH CATH Status
A 07 Apr, 2019 Chopped

CATH Domains (1)

Domain ID Date inserted into CATH Superfamily CATH Status
6mauA01 08 Apr, 2019 1.20.920.10 Assigned

UniProtKB Entries (1)

Accession Gene ID Taxon Description
O60885 BRD4_HUMAN Homo sapiens Bromodomain-containing protein 4