PDB Information

PDB6IAR
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli BL21(DE3)
Gene SourceHomo sapiens
Primary Citation
Tricyclic Indazoles-A Novel Class of Selective Estrogen Receptor Degrader Antagonists.
Scott, J.S., Bailey, A., Buttar, D., Carbajo, R.J., Curwen, J., Davey, P.R.J., Davies, R.D.M., Degorce, S.L., Donald, C., Gangl, E., Greenwood, R., Groombridge, S.D., Johnson, T., Lamont, S., Lawson, M., Lister, A., Morrow, C.J., Moss, T.A., Pink, J.H., Polanski, R.
J.Med.Chem.
HeaderDna Binding Protein
Released2018-11-27
Resolution1.840
CATH Insert Date27 Jan, 2019

PDB Images (3)

PDB Prints

PDB Chains (1)

Chain ID Date inserted into CATH CATH Status
A 27 Jan, 2019 Chopped

CATH Domains (1)

Domain ID Date inserted into CATH Superfamily CATH Status
6iarA00 28 Jan, 2019 1.10.565.10 Assigned

UniProtKB Entries (1)

Accession Gene ID Taxon Description
P03372 ESR1_HUMAN Homo sapiens Estrogen receptor