PDB 6hd4
PDB Information
PDB | 6HD4 |
Method | X-RAY DIFFRACTION |
Host Organism | Baculovirus expression vector pFastBac1-HM |
Gene Source | Mus musculus |
Primary Citation | Discovery of Asciminib (ABL001), an Allosteric Inhibitor of the Tyrosine Kinase Activity of BCR-ABL1.
J. Med. Chem.
|
Header | Transferase |
Released | 2018-08-17 |
Resolution | 2.030 |
CATH Insert Date | 16 Dec, 2018 |
PDB Images (7)
PDB Prints
PDB Chains (2)
Chain ID | Date inserted into CATH | CATH Status |
---|---|---|
A | 16 Dec, 2018 | Chopped |
B | 16 Dec, 2018 | Chopped |
CATH Domains (4)
Domain ID | Date inserted into CATH | Superfamily | CATH Status |
---|---|---|---|
6hd4A01 | 28 Feb, 2019 | 3.30.200.20 | Assigned |
6hd4A02 | 28 Feb, 2019 | 1.10.510.10 | Assigned |
6hd4B01 | 28 Feb, 2019 | 3.30.200.20 | Assigned |
6hd4B02 | 28 Feb, 2019 | 1.10.510.10 | Assigned |
UniProtKB Entries (2)
Accession | Gene ID | Taxon | Description |
---|---|---|---|
P00520 | ABL1_MOUSE | Mus musculus | Tyrosine-protein kinase ABL1 |
P00520 | ABL1_MOUSE | Mus musculus | Tyrosine-protein kinase ABL1 |