PDB Information

PDB6GXA
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli
Gene SourceSchistosoma mansoni
Primary Citation
Synthesis, Crystallization Studies, and in vitro Characterization of Cinnamic Acid Derivatives as SmHDAC8 Inhibitors for the Treatment of Schistosomiasis.
Bayer, T., Chakrabarti, A., Lancelot, J., Shaik, T.B., Hausmann, K., Melesina, J., Schmidtkunz, K., Marek, M., Erdmann, F., Schmidt, M., Robaa, D., Romier, C., Pierce, R.J., Jung, M., Sippl, W.
ChemMedChem
HeaderHydrolase
Released2018-06-27
Resolution2.100
CATH Insert Date19 Aug, 2018

PDB Images (9)

PDB Prints

PDB Chains (4)

Chain ID Date inserted into CATH CATH Status
A 19 Aug, 2018 Chopped
B 19 Aug, 2018 Chopped
C 19 Aug, 2018 Chopped
D 19 Aug, 2018 Chopped

CATH Domains (4)

Domain ID Date inserted into CATH Superfamily CATH Status
6gxaA00 20 Aug, 2018 3.40.800.20 Assigned
6gxaB00 20 Aug, 2018 3.40.800.20 Assigned
6gxaC00 20 Aug, 2018 3.40.800.20 Assigned
6gxaD00 20 Aug, 2018 3.40.800.20 Assigned

UniProtKB Entries (4)

Accession Gene ID Taxon Description
A5H660 A5H660_SCHMA Schistosoma mansoni Histone deacetylase 8
A5H660 A5H660_SCHMA Schistosoma mansoni Histone deacetylase 8
A5H660 A5H660_SCHMA Schistosoma mansoni Histone deacetylase 8
A5H660 A5H660_SCHMA Schistosoma mansoni Histone deacetylase 8