PDB Information

PDB6FX0
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli
Gene SourceHomo sapiens
Primary Citation
Structure-based design of Trifarotene (CD5789), a potent and selective RAR gamma agonist for the treatment of acne.
Thoreau, E., Arlabosse, J.M., Bouix-Peter, C., Chambon, S., Chantalat, L., Daver, S., Dumais, L., Duvert, G., Feret, A., Ouvry, G., Pascau, J., Raffin, C., Rodeville, N., Soulet, C., Tabet, S., Talano, S., Portal, T.
Bioorg. Med. Chem. Lett.
HeaderSignaling Protein
Released2018-03-08
Resolution1.900
CATH Insert Date03 Jun, 2018

PDB Images (3)

PDB Prints

PDB Chains (1)

Chain ID Date inserted into CATH CATH Status
A 03 Jun, 2018 Chopped

CATH Domains (1)

Domain ID Date inserted into CATH Superfamily CATH Status
6fx0A00 29 Jun, 2018 1.10.565.10 Assigned

UniProtKB Entries (1)

Accession Gene ID Taxon Description
P13631 RARG_HUMAN Homo sapiens Retinoic acid receptor gamma