PDB Information

PDB6E4F
MethodX-RAY DIFFRACTION
Host OrganismSpodoptera frugiperda
Gene SourceHomo sapiens
Primary Citation
The BTK Inhibitor ARQ 531 Targets Ibrutinib-Resistant CLL and Richter Transformation.
Reiff, S.D., Mantel, R., Smith, L.L., Greene, J.T., Muhowski, E.M., Fabian, C.A., Goettl, V.M., Tran, M., Harrington, B.K., Rogers, K.A., Awan, F.T., Maddocks, K., Andritsos, L., Lehman, A.M., Sampath, D., Lapalombella, R., Eathiraj, S., Abbadessa, G., Schwartz, B., Johnson, A.J., Byrd, J.C., Woyach, J.A.
Cancer Discov
HeaderSignaling Protein/Inhibitor
Released2018-07-17
Resolution1.150
CATH Insert Date09 Sep, 2018

PDB Images (4)

PDB Prints

PDB Chains (1)

Chain ID Date inserted into CATH CATH Status
A 09 Sep, 2018 Chopped

CATH Domains (2)

Domain ID Date inserted into CATH Superfamily CATH Status
6e4fA01 10 Sep, 2018 3.30.200.20 Assigned
6e4fA02 10 Sep, 2018 1.10.510.10 Assigned

UniProtKB Entries (1)

Accession Gene ID Taxon Description
Q06187 BTK_HUMAN Homo sapiens Tyrosine-protein kinase BTK