PDB Information

PDB6DGT
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli
Gene SourceMus musculus
Primary Citation
Atropisomerism by Design: Discovery of a Selective and Stable Phosphoinositide 3-Kinase (PI3K) beta Inhibitor.
Chandrasekhar, J., Dick, R., Van Veldhuizen, J., Koditek, D., Lepist, E.I., McGrath, M.E., Patel, L., Phillips, G., Sedillo, K., Somoza, J.R., Therrien, J., Till, N.A., Treiberg, J., Villasenor, A.G., Zherebina, Y., Perreault, S.
J. Med. Chem.
HeaderTransferase/Transferase Inhibitor
Released2018-05-18
Resolution2.600
CATH Insert Date05 Aug, 2018

PDB Images (2)

PDB Prints

PDB Chains (1)

Chain ID Date inserted into CATH CATH Status
A 05 Aug, 2018 Holding pen

CATH Domains (0)

Domain ID Date inserted into CATH Superfamily CATH Status

UniProtKB Entries (1)

Accession Gene ID Taxon Description
O35904 PK3CD_MOUSE Mus musculus Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform