PDB 6c4d
PDB Information
PDB | 6C4D |
Method | X-RAY DIFFRACTION |
Host Organism | Spodoptera frugiperda |
Gene Source | Homo sapiens |
Primary Citation | Discovery of 7-Oxo-2,4,5,7-tetrahydro-6 H-pyrazolo[3,4- c]pyridine Derivatives as Potent, Orally Available, and Brain-Penetrating Receptor Interacting Protein 1 (RIP1) Kinase Inhibitors: Analysis of Structure-Kinetic Relationships.
J. Med. Chem.
|
Header | Transferase/Transferase Inhibitor |
Released | 2018-01-11 |
Resolution | 2.520 |
CATH Insert Date | 03 Jun, 2018 |
PDB Images (13)
PDB Prints
PDB Chains (4)
Chain ID | Date inserted into CATH | CATH Status |
---|---|---|
A | 03 Jun, 2018 | Chopped |
B | 03 Jun, 2018 | Chopped |
C | 03 Jun, 2018 | Chopped |
D | 03 Jun, 2018 | Chopped |
CATH Domains (8)
Domain ID | Date inserted into CATH | Superfamily | CATH Status |
---|---|---|---|
6c4dA01 | 28 Jun, 2018 | 3.30.200.20 | Assigned |
6c4dA02 | 28 Jun, 2018 | 1.10.510.10 | Assigned |
6c4dB01 | 28 Jun, 2018 | 3.30.200.20 | Assigned |
6c4dB02 | 28 Jun, 2018 | 1.10.510.10 | Assigned |
6c4dC01 | 28 Jun, 2018 | 3.30.200.20 | Assigned |
6c4dC02 | 28 Jun, 2018 | 1.10.510.10 | Assigned |
6c4dD01 | 28 Jun, 2018 | 3.30.200.20 | Assigned |
6c4dD02 | 28 Jun, 2018 | 1.10.510.10 | Assigned |
UniProtKB Entries (4)
Accession | Gene ID | Taxon | Description |
---|---|---|---|
Q13546 | RIPK1_HUMAN | Homo sapiens | Receptor-interacting serine/threonine-protein kinase 1 |
Q13546 | RIPK1_HUMAN | Homo sapiens | Receptor-interacting serine/threonine-protein kinase 1 |
Q13546 | RIPK1_HUMAN | Homo sapiens | Receptor-interacting serine/threonine-protein kinase 1 |
Q13546 | RIPK1_HUMAN | Homo sapiens | Receptor-interacting serine/threonine-protein kinase 1 |