PDB Information

PDB6BSK
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli
Gene SourceHomo sapiens
Primary Citation
Discovery of 2,6-disubstituted pyrazine derivatives as inhibitors of CK2 and PIM kinases.
Gingipalli, L., Block, M.H., Bao, L., Cooke, E., Dakin, L.A., Denz, C.R., Ferguson, A.D., Johannes, J.W., Larsen, N.A., Lyne, P.D., Pontz, T.W., Wang, T., Wu, X., Wu, A., Zhang, H.J., Zheng, X., Dowling, J.E., Lamb, M.L.
Bioorg. Med. Chem. Lett.
HeaderTransferase/Transferase Inhibitor
Released2017-12-03
Resolution2.570
CATH Insert Date03 Jun, 2018

PDB Images (4)

PDB Prints

PDB Chains (1)

Chain ID Date inserted into CATH CATH Status
A 03 Jun, 2018 Chopped

CATH Domains (2)

Domain ID Date inserted into CATH Superfamily CATH Status
6bskA01 28 Jun, 2018 3.30.200.20 Assigned
6bskA02 28 Jun, 2018 1.10.510.10 Assigned

UniProtKB Entries (1)

Accession Gene ID Taxon Description
P11309 PIM1_HUMAN Homo sapiens Serine/threonine-protein kinase pim-1