PDB Information

PDB6B2P
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli
Gene SourceMycobacterium tuberculosis
Primary Citation
Mtb PKNA/PKNB Dual Inhibition Provides Selectivity Advantages for Inhibitor Design To Minimize Host Kinase Interactions.
Wang, T., Bemis, G., Hanzelka, B., Zuccola, H., Wynn, M., Moody, C.S., Green, J., Locher, C., Liu, A., Gao, H., Xu, Y., Wang, S., Wang, J., Bennani, Y.L., Thomson, J.A., Muh, U.
ACS Med Chem Lett
HeaderTransferase/Inhibitor
Released2017-09-20
Resolution3.010
CATH Insert Date03 Jun, 2018

PDB Images (4)

PDB Prints

PDB Chains (1)

Chain ID Date inserted into CATH CATH Status
A 03 Jun, 2018 Chopped

CATH Domains (2)

Domain ID Date inserted into CATH Superfamily CATH Status
6b2pA01 28 Jun, 2018 3.30.200.20 Assigned
6b2pA02 28 Jun, 2018 1.10.510.10 Assigned

UniProtKB Entries (1)

Accession Gene ID Taxon Description
P9WI81 PKNB_MYCTU Mycobacterium tuberculosis H37Rv Serine/threonine-protein kinase PknB