PDB Information

PDB6AXQ
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli
Gene SourceHomo sapiens
Primary Citation
A Unique Approach to Design Potent and Selective Cyclic Adenosine Monophosphate Response Element Binding Protein, Binding Protein (CBP) Inhibitors.
Bronner, S.M., Murray, J., Romero, F.A., Lai, K.W., Tsui, V., Cyr, P., Beresini, M.H., de Leon Boenig, G., Chen, Z., Choo, E.F., Clark, K.R., Crawford, T.D., Jayaram, H., Kaufman, S., Li, R., Li, Y., Liao, J., Liang, X., Liu, W., Ly, J., Maher, J., Wai, J., Wang, F., Zheng, A., Zhu, X., Magnuson, S.
J. Med. Chem.
HeaderTransferase/Transferase Inhibitor
Released2017-09-07
Resolution1.300
CATH Insert Date03 Jun, 2018

PDB Images (9)

PDB Prints

PDB Chains (4)

Chain ID Date inserted into CATH CATH Status
A 03 Jun, 2018 Chopped
B 03 Jun, 2018 Chopped
C 03 Jun, 2018 Chopped
D 03 Jun, 2018 Chopped

CATH Domains (4)

Domain ID Date inserted into CATH Superfamily CATH Status
6axqA00 28 Jun, 2018 1.20.920.10 Assigned
6axqB00 28 Jun, 2018 1.20.920.10 Assigned
6axqC00 28 Jun, 2018 1.20.920.10 Assigned
6axqD00 28 Jun, 2018 1.20.920.10 Assigned

UniProtKB Entries (4)

Accession Gene ID Taxon Description
Q92793 CBP_HUMAN Homo sapiens CREB-binding protein
Q92793 CBP_HUMAN Homo sapiens CREB-binding protein
Q92793 CBP_HUMAN Homo sapiens CREB-binding protein
Q92793 CBP_HUMAN Homo sapiens CREB-binding protein