PDB Information

PDB6AUD
MethodX-RAY DIFFRACTION
Host OrganismSpodoptera frugiperda
Gene SourceHomo sapiens
Primary Citation
Design of Selective Benzoxazepin PI3K delta Inhibitors Through Control of Dihedral Angles.
Safina, B.S., Elliott, R.L., Forrest, A.K., Heald, R.A., Murray, J.M., Nonomiya, J., Pang, J., Salphati, L., Seward, E.M., Staben, S.T., Ultsch, M., Wei, B., Yang, W., Sutherlin, D.P.
ACS Med Chem Lett
HeaderTransferase/Transferase Inhbitor
Released2017-08-31
Resolution2.020
CATH Insert Date17 Dec, 2017

PDB Images (7)

PDB Prints

PDB Chains (1)

Chain ID Date inserted into CATH CATH Status
A 17 Dec, 2017 Chopped

CATH Domains (5)

Domain ID Date inserted into CATH Superfamily CATH Status
6audA01 23 Dec, 2017 3.10.20.90 Assigned
6audA02 23 Dec, 2017 2.60.40.150 Assigned
6audA03 23 Dec, 2017 1.25.40.70 Assigned
6audA04 23 Dec, 2017 3.30.1010.10 Assigned
6audA05 23 Dec, 2017 1.10.1070.11 Assigned

UniProtKB Entries (1)

Accession Gene ID Taxon Description
P48736 PK3CG_HUMAN Homo sapiens Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform