PDB Information

PDB6AFR
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli K-12
Gene SourceHomo sapiens
Primary Citation
Rational design of 5-((1H-imidazol-1-yl)methyl)quinolin-8-ol derivatives as novel bromodomain-containing protein 4 inhibitors
Xing, J., Zhang, R., Jiang, X., Hu, T., Wang, X., Qiao, G., Wang, J., Yang, F., Luo, X., Chen, K., Shen, J., Luo, C., Jiang, H., Zheng, M.
Eur J Med Chem
HeaderSignaling Protein/Inhibitor
Released2018-08-08
Resolution2.000
CATH Insert Date16 Dec, 2018

PDB Images (3)

PDB Prints

PDB Chains (1)

Chain ID Date inserted into CATH CATH Status
A 16 Dec, 2018 Chopped

CATH Domains (1)

Domain ID Date inserted into CATH Superfamily CATH Status
6afrA01 28 Feb, 2019 1.20.920.10 Assigned

UniProtKB Entries (1)

Accession Gene ID Taxon Description
O60885 BRD4_HUMAN Homo sapiens Bromodomain-containing protein 4