PDB Information

PDB6A3N
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli BL21
Gene SourceHomo sapiens
Primary Citation
Discovery of Potent, Selective, and Orally Bioavailable Inhibitors against Phosphodiesterase-9, a Novel Target for the Treatment of Vascular Dementia.
Wu, Y., Zhou, Q., Zhang, T., Li, Z., Chen, Y.P., Zhang, P., Yu, Y.F., Geng, H., Tian, Y.J., Zhang, C., Wang, Y., Chen, J.W., Chen, Y., Luo, H.B.
J. Med. Chem.
HeaderHydrolase
Released2018-06-15
Resolution2.600
CATH Insert Date14 Apr, 2019

PDB Images (5)

PDB Prints

PDB Chains (2)

Chain ID Date inserted into CATH CATH Status
A 14 Apr, 2019 Chopped
B 14 Apr, 2019 Chopped

CATH Domains (2)

Domain ID Date inserted into CATH Superfamily CATH Status
6a3nA00 15 Apr, 2019 1.10.1300.10 Assigned
6a3nB00 15 Apr, 2019 1.10.1300.10 Assigned

UniProtKB Entries (2)

Accession Gene ID Taxon Description
O76083 PDE9A_HUMAN Homo sapiens High affinity cGMP-specific 3',5'-cyclic phosphodiesterase 9A
O76083 PDE9A_HUMAN Homo sapiens High affinity cGMP-specific 3',5'-cyclic phosphodiesterase 9A