PDB Information

PDB5YOJ
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli
Gene SourceHuman immunodeficiency virus 1
Primary Citation
Identification of Highly Potent Human Immunodeficiency Virus Type-1 Protease Inhibitors against Lopinavir and Darunavir Resistant Viruses from Allophenylnorstatine-Based Peptidomimetics with P2 Tetrahydrofuranylglycine.
Hidaka, K., Kimura, T., Sankaranarayanan, R., Wang, J., McDaniel, K.F., Kempf, D.J., Kameoka, M., Adachi, M., Kuroki, R., Nguyen, J.T., Hayashi, Y., Kiso, Y.
J. Med. Chem.
HeaderHydrolase/Hydrolase Inhibitor
Released2017-10-29
Resolution1.500
CATH Insert Date16 Jul, 2018

PDB Images (5)

PDB Prints

PDB Chains (2)

Chain ID Date inserted into CATH CATH Status
A 16 Jul, 2018 Chopped
B 16 Jul, 2018 Chopped

CATH Domains (2)

Domain ID Date inserted into CATH Superfamily CATH Status
5yojA00 19 Jul, 2018 2.40.70.10 Assigned
5yojB00 19 Jul, 2018 2.40.70.10 Assigned

UniProtKB Entries (2)

Accession Gene ID Taxon Description
P03366 POL_HV1B1 Human immunodeficiency virus type 1 BH10 Gag-Pol polyprotein
P03366 POL_HV1B1 Human immunodeficiency virus type 1 BH10 Gag-Pol polyprotein