PDB Information

PDB5Y9L
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli
Gene SourceHomo sapiens
Primary Citation
Discovery and structure-activity relationship study of 1,3,6-trisubstituted 1,4-diazepane-7-ones as novel human kallikrein 7 inhibitors
Murafuji, H., Sakai, H., Goto, M., Imajo, S., Sugawara, H., Muto, T.
Bioorg. Med. Chem. Lett.
HeaderHydrolase
Released2017-08-25
Resolution2.150
CATH Insert Date17 Dec, 2017

PDB Images (4)

PDB Prints

PDB Chains (1)

Chain ID Date inserted into CATH CATH Status
A 17 Dec, 2017 Chopped

CATH Domains (2)

Domain ID Date inserted into CATH Superfamily CATH Status
5y9lA01 23 Dec, 2017 Holding pen
5y9lA02 23 Dec, 2017 2.40.10.10 Assigned

UniProtKB Entries (1)

Accession Gene ID Taxon Description
P49862 KLK7_HUMAN Homo sapiens Kallikrein-7