PDB 5w4w

PDB Information

PDB5W4W
MethodX-RAY DIFFRACTION
Host OrganismInsect cell expression vector pTIE1
Gene SourceHomo sapiens
Primary Citation
Identification and Profiling of a Selective and Brain Penetrant Radioligand for in Vivo Target Occupancy Measurement of Casein Kinase 1 (CK1) Inhibitors.
Wager, T.T., Galatsis, P., Chandrasekaran, R.Y., Butler, T.W., Li, J., Zhang, L., Mente, S., Subramanyam, C., Liu, S., Doran, A.C., Chang, C., Fisher, K., Grimwood, S., Hedde, J.R., Marconi, M., Schildknegt, K.
ACS Chem Neurosci
HeaderTransferase/Inhibitor
Released2017-06-13
Resolution1.990
CATH Insert Date14 Nov, 2017

PDB Images (13)

PDB Prints

PDB Chains (4)

Chain ID Date inserted into CATH CATH Status
A 14 Nov, 2017 Chopped
B 14 Nov, 2017 Chopped
C 14 Nov, 2017 Chopped
D 14 Nov, 2017 Chopped

CATH Domains (8)

Domain ID Date inserted into CATH Superfamily CATH Status
5w4wA01 10 Dec, 2017 3.30.200.20 Assigned
5w4wA02 10 Dec, 2017 1.10.510.10 Assigned
5w4wB01 10 Dec, 2017 3.30.200.20 Assigned
5w4wB02 10 Dec, 2017 1.10.510.10 Assigned
5w4wC01 10 Dec, 2017 3.30.200.20 Assigned
5w4wC02 10 Dec, 2017 1.10.510.10 Assigned
5w4wD01 10 Dec, 2017 3.30.200.20 Assigned
5w4wD02 10 Dec, 2017 1.10.510.10 Assigned

UniProtKB Entries (4)

Accession Gene ID Taxon Description
P48730 KC1D_HUMAN Homo sapiens Casein kinase I isoform delta
P48730 KC1D_HUMAN Homo sapiens Casein kinase I isoform delta
P48730 KC1D_HUMAN Homo sapiens Casein kinase I isoform delta
P48730 KC1D_HUMAN Homo sapiens Casein kinase I isoform delta