PDB 5vom

PDB Information

PDB5VOM
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli
Gene SourceHomo sapiens
Primary Citation
Design and Optimization of Benzopiperazines as Potent Inhibitors of BET Bromodomains.
Millan, D.S., Kayser-Bricker, K.J., Martin, M.W., Talbot, A.C., Schiller, S.E.R., Herbertz, T., Williams, G.L., Luke, G.P., Hubbs, S., Alvarez Morales, M.A., Cardillo, D., Troccolo, P., Mendes, R.L., McKinnon, C.
ACS Med Chem Lett
HeaderTranscription/Inhibitor
Released2017-05-03
Resolution1.670
CATH Insert Date14 Nov, 2017

PDB Images (5)

PDB Prints

PDB Chains (2)

Chain ID Date inserted into CATH CATH Status
A 14 Nov, 2017 Chopped
B 14 Nov, 2017 Chopped

CATH Domains (2)

Domain ID Date inserted into CATH Superfamily CATH Status
5vomA01 10 Dec, 2017 1.20.920.10 Assigned
5vomB01 10 Dec, 2017 1.20.920.10 Assigned

UniProtKB Entries (2)

Accession Gene ID Taxon Description
O60885 BRD4_HUMAN Homo sapiens Bromodomain-containing protein 4
O60885 BRD4_HUMAN Homo sapiens Bromodomain-containing protein 4