PDB Information

PDB5VFD
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli
Gene SourceAcinetobacter baumannii
Primary Citation
ETX2514 is a broad-spectrum beta-lactamase inhibitor for the treatment of drug-resistant Gram-negative bacteria including Acinetobacter baumannii.
Durand-Reville, T.F., Guler, S., Comita-Prevoir, J., Chen, B., Bifulco, N., Huynh, H., Lahiri, S., Shapiro, A.B., McLeod, S.M., Carter, N.M., Moussa, S.H., Velez-Vega, C., Olivier, N.B., McLaughlin, R., Gao, N., Thresher, J., Palmer, T., Andrews, B., Giacobbe, R.A., Newman, J.V., Ehmann, D.E., de Jonge, B., O'Donnell, J., Mueller, J.P., Tommasi, R.A., Miller, A.A.
Nat Microbiol
HeaderHydrolase/Hydrolase Inhibitor
Released2017-04-07
Resolution1.930
CATH Insert Date14 Nov, 2017

PDB Images (3)

PDB Prints

PDB Chains (1)

Chain ID Date inserted into CATH CATH Status
A 14 Nov, 2017 Chopped

CATH Domains (1)

Domain ID Date inserted into CATH Superfamily CATH Status
5vfdA00 10 Dec, 2017 3.40.710.10 Assigned

UniProtKB Entries (1)

Accession Gene ID Taxon Description
Q8RLA6 Q8RLA6_ACIBA Acinetobacter baumannii Beta-lactamase