PDB Information

PDB5V5N
MethodX-RAY DIFFRACTION
Host OrganismSpodoptera frugiperda
Gene SourceHomo sapiens
Primary Citation
Takinib, a Selective TAK1 Inhibitor, Broadens the Therapeutic Efficacy of TNF-alpha Inhibition for Cancer and Autoimmune Disease.
Totzke, J., Gurbani, D., Raphemot, R., Hughes, P.F., Bodoor, K., Carlson, D.A., Loiselle, D.R., Bera, A.K., Eibschutz, L.S., Perkins, M.M., Eubanks, A.L., Campbell, P.L., Fox, D.A., Westover, K.D., Haystead, T.A.J., Derbyshire, E.R.
Cell Chem Biol
HeaderTransferase/Transferase Inhibitor
Released2017-03-14
Resolution2.010
CATH Insert Date14 Nov, 2017

PDB Images (4)

PDB Prints

PDB Chains (1)

Chain ID Date inserted into CATH CATH Status
A 14 Nov, 2017 Chopped

CATH Domains (2)

Domain ID Date inserted into CATH Superfamily CATH Status
5v5nA01 10 Dec, 2017 3.30.200.20 Assigned
5v5nA02 10 Dec, 2017 1.10.510.10 Assigned

UniProtKB Entries (2)

Accession Gene ID Taxon Description
O43318 M3K7_HUMAN Homo sapiens Mitogen-activated protein kinase kinase kinase 7
Q15750 TAB1_HUMAN Homo sapiens TGF-beta-activated kinase 1 and MAP3K7-binding protein 1