PDB Information

PDB5UWN
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli BL21(DE3)
Gene SourceHomo sapiens
Primary Citation
Structure-Based Design and Synthesis of Potent and Selective Matrix Metalloproteinase 13 Inhibitors.
Choi, J.Y., Fuerst, R., Knapinska, A.M., Taylor, A.B., Smith, L., Cao, X., Hart, P.J., Fields, G.B., Roush, W.R.
J. Med. Chem.
HeaderHydrolase/Hydrolase Inhibitor
Released2017-02-21
Resolution3.200
CATH Insert Date14 Nov, 2017

PDB Images (11)

PDB Prints

PDB Chains (5)

Chain ID Date inserted into CATH CATH Status
A 14 Nov, 2017 Chopped
B 14 Nov, 2017 Chopped
C 14 Nov, 2017 Chopped
D 14 Nov, 2017 Chopped
E 14 Nov, 2017 Chopped

CATH Domains (5)

Domain ID Date inserted into CATH Superfamily CATH Status
5uwnA00 10 Dec, 2017 3.40.390.10 Assigned
5uwnB00 10 Dec, 2017 3.40.390.10 Assigned
5uwnC00 10 Dec, 2017 3.40.390.10 Assigned
5uwnD00 10 Dec, 2017 3.40.390.10 Assigned
5uwnE00 10 Dec, 2017 3.40.390.10 Assigned

UniProtKB Entries (5)

Accession Gene ID Taxon Description
P45452 MMP13_HUMAN Homo sapiens Collagenase 3
P45452 MMP13_HUMAN Homo sapiens Collagenase 3
P45452 MMP13_HUMAN Homo sapiens Collagenase 3
P45452 MMP13_HUMAN Homo sapiens Collagenase 3
P45452 MMP13_HUMAN Homo sapiens Collagenase 3