PDB 5ur1
PDB Information
PDB | 5UR1 |
Method | X-RAY DIFFRACTION |
Host Organism | Escherichia coli |
Gene Source | Homo sapiens |
Primary Citation | 2-Oxo-3, 4-dihydropyrimido[4, 5-d]pyrimidinyl derivatives as new irreversible pan fibroblast growth factor receptor (FGFR) inhibitors.
Eur J Med Chem
|
Header | Transferase/Transferase Inhibitor |
Released | 2017-02-09 |
Resolution | 2.200 |
CATH Insert Date | 14 Nov, 2017 |
PDB Images (7)
PDB Prints
PDB Chains (2)
Chain ID | Date inserted into CATH | CATH Status |
---|---|---|
A | 14 Nov, 2017 | Chopped |
B | 14 Nov, 2017 | Chopped |
CATH Domains (4)
Domain ID | Date inserted into CATH | Superfamily | CATH Status |
---|---|---|---|
5ur1A01 | 10 Dec, 2017 | 3.30.200.20 | Assigned |
5ur1A02 | 10 Dec, 2017 | 1.10.510.10 | Assigned |
5ur1B01 | 10 Dec, 2017 | 3.30.200.20 | Assigned |
5ur1B02 | 10 Dec, 2017 | 1.10.510.10 | Assigned |
UniProtKB Entries (2)
Accession | Gene ID | Taxon | Description |
---|---|---|---|
P11362 | FGFR1_HUMAN | Homo sapiens | Fibroblast growth factor receptor 1 |
P11362 | FGFR1_HUMAN | Homo sapiens | Fibroblast growth factor receptor 1 |