PDB Information

PDB5TIU
MethodX-RAY DIFFRACTION
Host OrganismSpodoptera frugiperda
Gene SourceHomo sapiens
Primary Citation
Carboxamide Spleen Tyrosine Kinase (Syk) Inhibitors: Leveraging Ground State Interactions To Accelerate Optimization.
Ellis, J.M., Altman, M.D., Cash, B., Haidle, A.M., Kubiak, R.L., Maddess, M.L., Yan, Y., Northrup, A.B.
ACS Med Chem Lett
HeaderTransferase/Transferase Inhibitor
Released2016-10-03
Resolution1.490
CATH Insert Date07 May, 2017

PDB Images (4)

PDB Prints

PDB Chains (1)

Chain ID Date inserted into CATH CATH Status
A 08 May, 2017 Chopped

CATH Domains (2)

Domain ID Date inserted into CATH Superfamily CATH Status
5tiuA01 21 May, 2017 3.30.200.20 Assigned
5tiuA02 21 May, 2017 1.10.510.10 Assigned

UniProtKB Entries (1)

Accession Gene ID Taxon Description
P43405 KSYK_HUMAN Homo sapiens Tyrosine-protein kinase SYK