PDB Information

PDB5T23
MethodX-RAY DIFFRACTION
Host OrganismInsect cell expression vector pTIE1
Gene SourceHomo sapiens
Primary Citation
Discovery of triazole aminopyrazines as a highly potent and selective series of PI3K delta inhibitors.
Terstiege, I., Perry, M., Petersen, J., Tyrchan, C., Svensson, T., Lindmark, H., Oster, L.
Bioorg. Med. Chem. Lett.
HeaderTransferase
Released2016-08-23
Resolution2.780
CATH Insert Date07 May, 2017

PDB Images (7)

PDB Prints

PDB Chains (1)

Chain ID Date inserted into CATH CATH Status
A 08 May, 2017 Chopped

CATH Domains (5)

Domain ID Date inserted into CATH Superfamily CATH Status
5t23A01 20 May, 2017 3.10.20.90 Assigned
5t23A02 20 May, 2017 2.60.40.150 Assigned
5t23A03 20 May, 2017 1.25.40.70 Assigned
5t23A04 20 May, 2017 3.30.1010.10 Assigned
5t23A05 20 May, 2017 1.10.1070.11 Assigned

UniProtKB Entries (1)

Accession Gene ID Taxon Description
P48736 PK3CG_HUMAN Homo sapiens Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform