PDB Information

PDB5OW8
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli BL21(DE3)
Gene SourceHomo sapiens
Primary Citation
Discovery of a Series of Indole-2 Carboxamides as Selective Secreted Phospholipase A2Type X (sPLA2-X) Inhibitors.
Knerr, L., Giordanetto, F., Nordberg, P., Pettersen, D., Selmi, N., Beisel, H.G., de la Motte, H., Olsson, T., Perkins, T.D.J., Herslof, M., Mansson, A., Dahlstrom, M., Starke, I., Broddefalk, J., Saarinen, G., Klingegard, F., Hurt-Camejo, E., Rosengren, B., Brengdahl, J., Jansen, F., Rohman, M., Sandmark, J., Hallberg, K., Akerud, T., Roth, R.G., Ahlqvist, M.
ACS Med Chem Lett
HeaderLipid Binding Protein
Released2017-08-31
Resolution1.900
CATH Insert Date05 Aug, 2018

PDB Images (5)

PDB Prints

PDB Chains (2)

Chain ID Date inserted into CATH CATH Status
A 05 Aug, 2018 Chopped
B 05 Aug, 2018 Chopped

CATH Domains (2)

Domain ID Date inserted into CATH Superfamily CATH Status
5ow8A00 06 Aug, 2018 1.20.90.10 Assigned
5ow8B00 06 Aug, 2018 1.20.90.10 Assigned

UniProtKB Entries (2)

Accession Gene ID Taxon Description
O15496 PA2GX_HUMAN Homo sapiens Group 10 secretory phospholipase A2
O15496 PA2GX_HUMAN Homo sapiens Group 10 secretory phospholipase A2