PDB Information

PDB5O7I
MethodX-RAY DIFFRACTION
Host OrganismSpodoptera frugiperda
Gene SourceHomo sapiens
Primary Citation
Identification of a novel orally bioavailable ERK5 inhibitor with selectivity over p38 alpha and BRD4.
Myers, S.M., Miller, D.C., Molyneux, L., Arasta, M., Bawn, R.H., Blackburn, T.J., Cook, S.J., Edwards, N., Endicott, J.A., Golding, B.T., Griffin, R.J., Hammonds, T., Hardcastle, I.R., Harnor, S.J., Heptinstall, A.B., Lochhead, P.A., Martin, M.P., Martin, N.C., Newell, D.R., Owen, P.J., Pang, L.C., Reuillon, T., Rigoreau, L.J.M., Thomas, H.D., Tucker, J.A., Wang, L.Z., Wong, A.C., Noble, M.E.M., Wedge, S.R., Cano, C.
Eur.J.Med.Chem.
HeaderTransferase
Released2017-06-08
Resolution2.380
CATH Insert Date06 Jul, 2018

PDB Images (2)

PDB Prints

PDB Chains (1)

Chain ID Date inserted into CATH CATH Status
A 06 Jul, 2018 Check for files

CATH Domains (0)

Domain ID Date inserted into CATH Superfamily CATH Status

UniProtKB Entries (0)

Accession Gene ID Taxon Description